A Targeted Small Molecule Approach to Essential Tremor

Developing DK-I-56-1, a differentiated GABA-A subtype-selective therapy designed to address the unmet need in essential tremor.

Primary Indication: Essential Tremor

Selective Mechanism: Cerebellar GABA-A subtype targeting

Development Stage: Preclinical

Partnering Strategy: Milestone-driven value creation

Essential Tremor

A common movement disorder characterized by involuntary shaking, most often affecting the hands during action and daily activities.

Action Tremor

Shaking worsens during purposeful movement and daily tasks.

Severe Quality-of-Life Impact

Writing, eating, and fine motor tasks become difficult or impossible.

Chronic, Progressive Burden

Symptoms often worsen over time, limiting independence.

Current Treatment Landscape

Approved therapies exist, but many patients remain inadequately controlled.

First-line treatment relies on beta-blockers and anticonvulsants.

Propranolol & Primidone as Standard of Care

Often limited by incomplete efficacy, side effects, or contraindications.

Market Opportunity

~7M

Patients in the United States

Significant commercial opportunity in essential tremor

Current Treatment Landscape

Propranolol & Primidone

  • FDA-approved first-line therapies
  • Broad CNS and systemic effects
  • Non-selective mechanism of action
  • Established but incomplete efficacy in many patients

Efficacy & Tolerability Limits

  • Fatigue, sedation, and bradycardia
  • Contraindications in asthma and heart disease
  • Many patients seek additional or alternative options

A substantial portion of essential tremor patients remain inadequately treated.

Significant unmet need for a selective, better-tolerated alternative.

The Asset

DK-I-56-1

DK-I-56-1

A novel small-molecule therapy designed to selectively modulate a rare GABA-A receptor subtype expressed in cerebellar circuits involved in tremor control.

  • Small-molecule neuromodulator
  • Targets a rare GABA-A receptor subtype
  • Designed for selective cerebellar circuit modulation

Selective Targeting

Designed to act on a rare GABA-A subtype rather than broadly affecting CNS receptors.

Improved Tolerability Potential

Selective modulation may reduce sedation and CNS side effects associated with existing therapies.

Preclinical Evidence

Demonstrated activity in validated preclinical models of tremor.

Development Strategy

A focused path to clinical value creation.

Head-to-Head Preclinical Study

Comparing DK-I-56-1 directly against standard-of-care therapies in validated tremor models.

Demonstrate Differentiation

Generate data supporting selective targeting and improved CNS tolerability.

Partner for Clinical Development

Advance toward licensing or strategic partnership following successful preclinical results.

Milestones and Use of Funds

The next value-creation phase.

600K Raise

Funding a focused preclinical validation program.

Head-to-Head Study

Execute preclinical comparison of DK-I-56-1 vs standard-of-care therapies.

Data Generation

Establish differentiation in efficacy and tolerability.

Business Development

Engage potential pharmaceutical partners.

Value Inflection

Position the program for licensing or strategic partnership.

A clear partnering milestone.

Generating the data needed to support strategic collaboration.

Traction & Credibility

Early validation from industry and research partners.

Pharma Collaboration

Prior development partnership with a major pharmaceutical company.

CRO Continuity

The same CRO team that advanced the previous program remains engaged.

Partner Interest

Early conversations with potential pharmaceutical partners.

Positioned for strategic partnership.

Focused execution with experienced collaborators.

Leadership Team

Experienced scientists advancing targeted neurological therapeutics.

Portrait of Michael Hendrickson

Michael Hendrickson

18 years in neuroscience & drug development; former Director of Preclinical Development and VP of Operations.

Portrait of Joseph Beck

Joseph Beck, PhD

Neuroscientist and serial entrepreneur with three successful startups.

Portrait of Barry Steiglitz

Barry Steiglitz, PhD

18 years pre-clinical research, including serving as principal investigator.

Portrait of Alex Kasper

Alex Kasper

20 years of CFO experience, including 14 years in small pharmaceutical companies.

Proven track record in neuroscience ventures.

The team previously partnered a small-molecule asset to MapLight Therapeutics, contributing to $600M in fundraising and a $300M IPO.

Ready to explore the opportunity?

NeuroSolis is advancing a differentiated preclinical therapy for essential tremor, targeting cerebellar circuits through selective GABA-A modulation.

For investor inquiries, partnering discussions, or access to additional diligence materials, contact the NeuroSolis team below.

  • Investor Inquiries
  • Partnering Discussions
  • Request Data Room Access